Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T6658 |
SB-408124
N-(6,8-二氟-2-甲基-4-喹啉)- N-[4-(二甲氨基)苯基]尿素 |
OX Receptor | GPCR/G Protein; Neuroscience |
SB408124 是一种 OX1 受体的非肽拮抗剂,在全细胞和膜中的 Ki 值分别为 57 和 27 nM,其选择性是 OX2 受体的 50 倍。 | |||
T12844 |
SB-408124 Hydrochloride
|
Others | Others |
SB-408124 Hydrochloride is a non-peptide OX1 receptor antagonist(Ki of 57 nM and 27 nM in both whole cell and membrane, respectively). |